Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists.

Saved in:
Bibliographic Details
Title: Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists.
Authors: Hintermann S; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Guntermann C; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Mattes H; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Carcache DA; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Wagner J; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Vulpetti A; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Billich A; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Dawson J; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Kaupmann K; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Kallen J; CPC, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Stringer R; MAP, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Orain D; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.
Source: ChemMedChem [ChemMedChem] 2016 Dec 16; Vol. 11 (24), pp. 2640-2648. Date of Electronic Publication: 2016 Nov 30.
Publication Type: Journal Article
Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE
Database: MEDLINE Ultimate
FullText Links:
  – Type: pdflink
Text:
  Availability: 0
Header DbId: mdl
DbLabel: MEDLINE Ultimate
An: 27902884
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AU" term="%22Hintermann+S%22">Hintermann S</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Guntermann+C%22">Guntermann C</searchLink>; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Mattes+H%22">Mattes H</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Carcache+DA%22">Carcache DA</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Wagner+J%22">Wagner J</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Vulpetti+A%22">Vulpetti A</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Billich+A%22">Billich A</searchLink>; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Dawson+J%22">Dawson J</searchLink>; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Kaupmann+K%22">Kaupmann K</searchLink>; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Kallen+J%22">Kallen J</searchLink>; CPC, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Stringer+R%22">Stringer R</searchLink>; MAP, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Orain+D%22">Orain D</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%22101259013%22">ChemMedChem</searchLink> [ChemMedChem] 2016 Dec 16; Vol. 11 (24), pp. 2640-2648. <i>Date of Electronic Publication: </i>2016 Nov 30.
– Name: TypePub
  Label: Publication Type
  Group: TypPub
  Data: Journal Article
– Name: TitleSource
  Label: Journal Info
  Group: Src
  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Wiley-VCH%22">Wiley-VCH </searchLink><i>Country of Publication: </i>Germany <i>NLM ID: </i>101259013 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1860-7187 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2218607179%22">18607179 </searchLink><i>NLM ISO Abbreviation: </i>ChemMedChem <i>Subsets: </i>MEDLINE
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=27902884
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1002/cmdc.201600500
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        StartPage: 2640
    Titles:
      – TitleFull: Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: Hintermann S
      – PersonEntity:
          Name:
            NameFull: Guntermann C
      – PersonEntity:
          Name:
            NameFull: Mattes H
      – PersonEntity:
          Name:
            NameFull: Carcache DA
      – PersonEntity:
          Name:
            NameFull: Wagner J
      – PersonEntity:
          Name:
            NameFull: Vulpetti A
      – PersonEntity:
          Name:
            NameFull: Billich A
      – PersonEntity:
          Name:
            NameFull: Dawson J
      – PersonEntity:
          Name:
            NameFull: Kaupmann K
      – PersonEntity:
          Name:
            NameFull: Kallen J
      – PersonEntity:
          Name:
            NameFull: Stringer R
      – PersonEntity:
          Name:
            NameFull: Orain D
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 16
              M: 12
              Text: 2016 Dec 16
              Type: published
              Y: 2016
          Identifiers:
            – Type: issn-electronic
              Value: 1860-7187
          Numbering:
            – Type: volume
              Value: 11
            – Type: issue
              Value: 24
          Titles:
            – TitleFull: ChemMedChem
              Type: main
ResultId 1