Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists.
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| Title: | Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists. |
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| Authors: | Hintermann S; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Guntermann C; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Mattes H; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Carcache DA; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Wagner J; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Vulpetti A; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Billich A; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Dawson J; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Kaupmann K; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Kallen J; CPC, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Stringer R; MAP, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland., Orain D; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland. |
| Source: | ChemMedChem [ChemMedChem] 2016 Dec 16; Vol. 11 (24), pp. 2640-2648. Date of Electronic Publication: 2016 Nov 30. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Links: – Type: pdflink Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 27902884 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Hintermann+S%22">Hintermann S</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Guntermann+C%22">Guntermann C</searchLink>; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Mattes+H%22">Mattes H</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Carcache+DA%22">Carcache DA</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Wagner+J%22">Wagner J</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Vulpetti+A%22">Vulpetti A</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Billich+A%22">Billich A</searchLink>; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Dawson+J%22">Dawson J</searchLink>; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Kaupmann+K%22">Kaupmann K</searchLink>; ATI, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Kallen+J%22">Kallen J</searchLink>; CPC, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Stringer+R%22">Stringer R</searchLink>; MAP, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland.<br /><searchLink fieldCode="AU" term="%22Orain+D%22">Orain D</searchLink>; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Novartis Campus, 4002, Basel, Switzerland. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101259013%22">ChemMedChem</searchLink> [ChemMedChem] 2016 Dec 16; Vol. 11 (24), pp. 2640-2648. <i>Date of Electronic Publication: </i>2016 Nov 30. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Wiley-VCH%22">Wiley-VCH </searchLink><i>Country of Publication: </i>Germany <i>NLM ID: </i>101259013 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1860-7187 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2218607179%22">18607179 </searchLink><i>NLM ISO Abbreviation: </i>ChemMedChem <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=27902884 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1002/cmdc.201600500 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 2640 Titles: – TitleFull: Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Hintermann S – PersonEntity: Name: NameFull: Guntermann C – PersonEntity: Name: NameFull: Mattes H – PersonEntity: Name: NameFull: Carcache DA – PersonEntity: Name: NameFull: Wagner J – PersonEntity: Name: NameFull: Vulpetti A – PersonEntity: Name: NameFull: Billich A – PersonEntity: Name: NameFull: Dawson J – PersonEntity: Name: NameFull: Kaupmann K – PersonEntity: Name: NameFull: Kallen J – PersonEntity: Name: NameFull: Stringer R – PersonEntity: Name: NameFull: Orain D IsPartOfRelationships: – BibEntity: Dates: – D: 16 M: 12 Text: 2016 Dec 16 Type: published Y: 2016 Identifiers: – Type: issn-electronic Value: 1860-7187 Numbering: – Type: volume Value: 11 – Type: issue Value: 24 Titles: – TitleFull: ChemMedChem Type: main |
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