Characterization of Specific N-α-Acetyltransferase 50 (Naa50) Inhibitors Identified Using a DNA Encoded Library.
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| Title: | Characterization of Specific N-α-Acetyltransferase 50 (Naa50) Inhibitors Identified Using a DNA Encoded Library. |
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| Authors: | Kung PP; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Bingham P; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Burke BJ; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Chen Q; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China., Cheng X; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China., Deng YL; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Dou D; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China., Feng J; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Gallego GM; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Gehring MR; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Grant SK; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Greasley S; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Harris AR; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Maegley KA; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Meier J; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Meng X; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China., Montano JL; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States., Morgan BA; HitGen Pharmaceuticals Inc., PO Box 88240, Houston, Texas 77288, United States.; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China., Naughton BS; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Palde PB; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Paul TA; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Richardson P; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Sakata S; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Shaginian A; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China., Sonnenburg WK; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China., Subramanyam C; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Timofeevski S; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Wan J; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China., Yan W; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States., Stewart AE; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States. |
| Source: | ACS medicinal chemistry letters [ACS Med Chem Lett] 2020 Apr 10; Vol. 11 (6), pp. 1175-1184. Date of Electronic Publication: 2020 Apr 10 (Print Publication: 2020). |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 32550998 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Characterization of Specific N-α-Acetyltransferase 50 (Naa50) Inhibitors Identified Using a DNA Encoded Library. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Kung+PP%22">Kung PP</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Bingham+P%22">Bingham P</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Burke+BJ%22">Burke BJ</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Chen+Q%22">Chen Q</searchLink>; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.<br /><searchLink fieldCode="AU" term="%22Cheng+X%22">Cheng X</searchLink>; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.<br /><searchLink fieldCode="AU" term="%22Deng+YL%22">Deng YL</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Dou+D%22">Dou D</searchLink>; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.<br /><searchLink fieldCode="AU" term="%22Feng+J%22">Feng J</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Gallego+GM%22">Gallego GM</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Gehring+MR%22">Gehring MR</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Grant+SK%22">Grant SK</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Greasley+S%22">Greasley S</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Harris+AR%22">Harris AR</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Maegley+KA%22">Maegley KA</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Meier+J%22">Meier J</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Meng+X%22">Meng X</searchLink>; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.<br /><searchLink fieldCode="AU" term="%22Montano+JL%22">Montano JL</searchLink>; Chemical Biology Laboratory, National Cancer Institute, Frederick, Maryland 21702, United States.<br /><searchLink fieldCode="AU" term="%22Morgan+BA%22">Morgan BA</searchLink>; HitGen Pharmaceuticals Inc., PO Box 88240, Houston, Texas 77288, United States.; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.<br /><searchLink fieldCode="AU" term="%22Naughton+BS%22">Naughton BS</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Palde+PB%22">Palde PB</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Paul+TA%22">Paul TA</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Richardson+P%22">Richardson P</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Sakata+S%22">Sakata S</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Shaginian+A%22">Shaginian A</searchLink>; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.<br /><searchLink fieldCode="AU" term="%22Sonnenburg+WK%22">Sonnenburg WK</searchLink>; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.<br /><searchLink fieldCode="AU" term="%22Subramanyam+C%22">Subramanyam C</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Timofeevski+S%22">Timofeevski S</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Wan+J%22">Wan J</searchLink>; HitGen Inc., Building 6, No.8, Huigu first East Road, Tianfu International Bio-Town, Shuangliu District, Chengdu, Sichuan 610200, P.R. China.<br /><searchLink fieldCode="AU" term="%22Yan+W%22">Yan W</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Stewart+AE%22">Stewart AE</searchLink>; Worldwide Research and Development, Pfizer Inc., 10770 Science Center Drive, San Diego, California 92121, United States. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101521073%22">ACS medicinal chemistry letters</searchLink> [ACS Med Chem Lett] 2020 Apr 10; Vol. 11 (6), pp. 1175-1184. <i>Date of Electronic Publication: </i>2020 Apr 10 (<i>Print Publication: </i>2020). – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101521073 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>1948-5875 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219485875%22">19485875 </searchLink><i>NLM ISO Abbreviation: </i>ACS Med Chem Lett <i>Subsets: </i>PubMed not MEDLINE |
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| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acsmedchemlett.0c00029 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 1175 Titles: – TitleFull: Characterization of Specific N-α-Acetyltransferase 50 (Naa50) Inhibitors Identified Using a DNA Encoded Library. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Kung PP – PersonEntity: Name: NameFull: Bingham P – PersonEntity: Name: NameFull: Burke BJ – PersonEntity: Name: NameFull: Chen Q – PersonEntity: Name: NameFull: Cheng X – PersonEntity: Name: NameFull: Deng YL – PersonEntity: Name: NameFull: Dou D – PersonEntity: Name: NameFull: Feng J – PersonEntity: Name: NameFull: Gallego GM – PersonEntity: Name: NameFull: Gehring MR – PersonEntity: Name: NameFull: Grant SK – PersonEntity: Name: NameFull: Greasley S – PersonEntity: Name: NameFull: Harris AR – PersonEntity: Name: NameFull: Maegley KA – PersonEntity: Name: NameFull: Meier J – PersonEntity: Name: NameFull: Meng X – PersonEntity: Name: NameFull: Montano JL – PersonEntity: Name: NameFull: Morgan BA – PersonEntity: Name: NameFull: Naughton BS – PersonEntity: Name: NameFull: Palde PB – PersonEntity: Name: NameFull: Paul TA – PersonEntity: Name: NameFull: Richardson P – PersonEntity: Name: NameFull: Sakata S – PersonEntity: Name: NameFull: Shaginian A – PersonEntity: Name: NameFull: Sonnenburg WK – PersonEntity: Name: NameFull: Subramanyam C – PersonEntity: Name: NameFull: Timofeevski S – PersonEntity: Name: NameFull: Wan J – PersonEntity: Name: NameFull: Yan W – PersonEntity: Name: NameFull: Stewart AE IsPartOfRelationships: – BibEntity: Dates: – D: 10 M: 04 Text: 2020 Apr 10 Type: published Y: 2020 Identifiers: – Type: issn-print Value: 1948-5875 Numbering: – Type: volume Value: 11 – Type: issue Value: 6 Titles: – TitleFull: ACS medicinal chemistry letters Type: main |
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